R590,00
Neuroprotection, Cognitive Enhancement, Memory, Learning Speed, Focus, Anti-Aging, Brain Support, Neuroinflammation, Strong Sleep Aid.
R590,00
9 in stock
Pinealon is a lab-made synthetic tripeptide – a super-short chain of just 3 amino acids (Glu-Asp-Arg) copied from natural proteins in the pineal gland and brain tissue. Developed in the 2000s by Russian scientist Prof. Vladimir Khavinson and his team as part of their ‘bioregulator’ peptide family, it is designed to target the central nervous system specifically. Unlike Epitalon (which focuses more on pineal melatonin and telomeres), Pinealon is the brain-specific version – tiny enough to cross cell and nuclear membranes and directly influence neuronal gene expression.
Think of Pinealon as your brain’s ‘cellular tune-up crew.’ It slips straight into neurons and flips protective gene switches.
How it works:
– Enters the nucleus and regulates gene expression for neuronal proteins.
– Suppresses free radicals (ROS), prevents apoptosis (cell death), and activates proliferative/repair pathways.
– Boosts neuron resilience to stress (oxidative, hypoxic, age-related).
– Neuroprotection: shields brain cells from oxidative damage, hypoxia, and age-related decline; improves neuron survival.
– Cognitive enhancement: better memory, learning speed, focus, and motor reactions (seen in monkey and rat studies).
– Anti-aging brain support: counters cognitive decline in elderly models; protects developing brains (e.g., prenatal stress).
– Possible circadian & mood signals: indirect pineal influence for better sleep-wake balance.
– Bonus hints: reduced neuroinflammation and improved recovery in vascular/traumatic brain issues.
In short: It helps your brain cells stay healthy, think sharper, and resist aging – like a targeted brain longevity switch.
Pinealon has one of the cleanest safety profiles among Khavinson peptides – decades of Russian use with almost no issues reported.
In available studies (preclinical + small human): No serious adverse events or organ toxicity.
Mild/rare effects:
– Injection-site redness or mild irritation.
– Occasional headache, dizziness, nausea, or temporary sleep changes (very uncommon).
Bigger caveats:
– Limited modern long-term Western data – most safety comes from short courses in elderly patients.
– Theoretical risk: any gene-modulating peptide could interact with existing conditions (though none reported).
Bottom line: Extremely well-tolerated in studied doses, but still experimental medical supervision recommended.
Method of Administration: Subcutaneous into fatty tissue.
Reconstitution: 2ml Bac water into single vial. See Reconstitution Guide
Dose: 2mg daily, therefore 20 units or 0.2ml. Use peptide calculator for alternative dosage.
Course: 20 days.
Cycling: Repeat every 3 months for maintenance or as needed (e.g., during respiratory seasons or after illness).
Tip: Reconstitute with bacteriostatic water; store in fridge. Use insulin syringes and sterile technique.
– Brain-specific bioregulator – the EDR tripeptide is tailored for neurons (while Epitalon is the pineal version).
– Nuclear passport – so small it crosses both cell and nuclear membranes to directly tweak gene expression.
– Monkey memory boost – in one study, macaques learned visual tasks much faster after just 10 days.
– Prenatal protector – helped rat pups born under stress develop better brains and motor skills.
– Khavinson family – one of over 20 short peptides he developed; all designed to ‘re-educate’ aging cells.
– Free-radical firefighter – one of the few peptides shown to lower ROS inside brain cells at very low doses.
– Russian longevity staple – used clinically in Russia for decades for age-related cognitive support.
Human data is limited (mostly small Russian observations and preclinical); large RCTs are still needed.
1. Innerbody Research (updated Jan 2026): Comprehensive review – neuroprotection, cognitive benefits, safety profile, and typical dosing.
2. Meshchaninov et al. (2015) Bulletin of Experimental Biology & Medicine: Pinealon + Vesugen in elderly with chronic brain syndrome – anabolic/neuroprotective effects, slowed biological aging, safe on genetic level.
3. Arutjunyan et al. (2012) International Journal of Clinical & Experimental Medicine: Pinealon protected rat offspring from prenatal hyperhomocysteinemia – improved cognition and neuron resistance to oxidative stress.
4. Khavinson et al. (2011) Rejuvenation Research: Pinealon increased cell viability by suppressing free radicals and activating proliferative processes in neurons.
5. Paragon Sports Medicine (2025-2026): Summary of 6+ studies showing cognitive enhancement, circadian regulation, neuroprotection; excellent tolerability.
6. Behemoth Labz (2025): Benefits, mechanism, and preclinical side-effect profile (minimal).
7. Biotech Peptides (20242026 updates): Neuroprotection in hypoxic models and gene-regulation mechanisms.
8. Core Peptides (20242026): Neuron protection, reduced ROS/necrosis, cognitive/motor benefits in prenatal and adult rat models.
9. Ilina et al. (2022) International Journal of Molecular Sciences (PMC): Ultrashort peptides like Pinealon as neuroprotective agents in Alzheimers models epigenetic mechanisms.
10. Recess RX / Peptides.org summaries (2026): Off-label cognitive & anti-aging uses; 1020 day cycle protocols.
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All products are sold in powder (lyophilized) form and require reconstitution with a suitable diluent for research purposes only. Research supplies (e.g., syringes, bacteriostatic water) are not included and need to be purchased separately. No personal human dosing instructions are provided, only research dosages from clinical studies. We adhere to all local and national (SAHPRA) laws around Research Only Chemical sales. We are not a pharmacy, nor do we promote or provide any advice for human or animal consumption. Please review our terms and conditions carefully before making a purchase on our website.
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